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Concentrations of naltrexone begin to slowly decline about 2 weeks after dosing, and levels of the medication stay measurable for a month or more. The elimination half life of naltrexone from Vivitrol ranges between 5 to 10 days.
You should tell your doctor if any of the following side effects become severe or don’t go away: Nausea, vomiting, diarrhea, or constipation. Stomach pain or cramping. Loss of appetite. Headache. Dizziness. Nervousness, irritability, or anxiety. Tearfulness. Increased or decreased energy.
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In terms of dosing, 50mg of naltrexone have the ability to block the effects of opioids for about 24 hours. Clinical studies suggest that doubling the dose will block opioid effects for 48 hours, while 150mg of naltrexone can provide blockage for approximately 72 hours. -
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