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Not to be confused with the related chemical naloxone. Naltrexone reverses the effects of opioids and is used primarily in the management of alcohol dependence and opioid dependence. It is marketed in generic form as its hydrochloride salt, naltrexone hydrochloride, and marketed under the trade names Revia and Depade.
What will happen if a patient drinks alcohol while taking naltrexone? Naltrexone does not reduce the effects of alcohol that impair coordination and judgment. Naltrexone may reduce the feeling of intoxication and the desire to drink more, but it will not cause a severe physical response to drinking. 5.
A dose of 50 mg once daily is recommended for most patients. The placebo-controlled studies that demonstrated the efficacy of Naltrexone hydrochloride tablets as an adjunctive treatment of alcoholism used a dose regimen of Naltrexone hydrochloride tablets 50 mg once daily for up to 12 weeks.
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The mean elimination half-life (T-?) values for naltrexone and 6-?-naltrexol are 4 hours and 13 hours, respectively. Naltrexone and 6-?-naltrexol are dose proportional in terms of AUC and Cmax over the range of 50 to 200 mg and do not accumulate after 100 mg daily doses. -
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